NPR1

NPR1

NPR1 Overview

Molecule Name
Natriuretic peptide receptor 1
Synonyms
Atrial natriuretic peptide receptor 1,NPR1,NPRA,GC-A,ANPRA,NPR-A
Drug Development Progress
Drugs in Clinical Trials7
Approved Drugs4
Highest Development StageApproved
Target Synonym
EC:4.6.1.2,Atrionatriuretic Peptide Receptor A,Natriuretic Peptide Receptor A,ANPRA,Atrial Natriuretic Peptide Receptor 1,Natriuretic Peptide A Type Receptor,Testicular Tissue Protein Li 20,EC 4.6.1.2,GUCY2A,GUC2A,ANPa,NPRA,GC-A,NPR-A,NPR1,Guanylate cyclase A,ANP-A,Natriuretic Peptide Receptor 1,Atrial Natriuretic Peptide Receptor Type A,ANPR-A,Natriuretic Peptide Receptor A/Guanylate Cyclase A (Atrionatriuretic Peptide Receptor A)
Background
Receptor for the atrial natriuretic peptide NPPA/ANP and the brain natriuretic peptide NPPB/BNP which are potent vasoactive hormones playing a key role in cardiovascular homeostasis. Has guanylate cyclase activity upon binding of the ligand.

NPR1 Product List

Species
  • Human(3)
  • Cynomolgus(1)
  • Mouse(1)
Tag
  • His Tag(3)
  • Fc Tag(1)
  • His Tag & Avi Tag(1)
Host
  • HEK293(5)
Conjugate
  • Unconjugated(4)
  • Biotin-labeled(1)
Grade
  • RUO(5)
Low Endotoxin
  • Yes(2)
  • No(3)
MoleculeCat. No.Product NameSpeciesHostStructurePurityActivitySize&Price
NPR1
HOTAvitag
NP1-H82E9
Biotinylated Human NPR1 / NPRA Protein, His,Avitag™ (MALS verified)
Human
HEK293
MALSSDS-PAGE
ELISA

$360.00

25ug
NPR1
Human NPR1 / NPRA Protein, Fc Tag (MALS verified)
Human
HEK293
MALSSDS-PAGE
ELISA

$430.00

100ug
NPR1
Mouse NPR1 / NPRA Protein, His Tag, low endotoxin (MALS verified)
Mouse
HEK293
MALSSDS-PAGE
ELISA

$395.00

100ug
NPR1
Cynomolgus NPR1 / NPRA Protein, His Tag, low endotoxin (MALS verified)
Cynomolgus
HEK293
MALSSDS-PAGE

$385.00

100ug
NPR1
Human NPR1 / NPRA Protein, His Tag (MALS verified)
Human
HEK293
MALSSDS-PAGE
ELISA

$385.00

100ug
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Clinical Drug Information

English NameResearch CodeHighest Development StageCompanyIndicationClinical Trial
Recombinant human brain natriuretic peptide(Shijiazhuang wotai)Phase 3 ClinicalShijiazhuang wotai Biotechnology Co Ltd
Acutely decompensated congestive heart failure; Heart Failure
Details
Recombinant human brain natriuretic peptide (Shanghai Jiao Tong University)Phase 3 ClinicalShanghai Jiaotong University
Heart Defects, Congenital; Tetralogy of Fallot
Details
NesiritideBNP-32 (human); JNS-004; hBNP; SC-70400Phase 2 ClinicalJohnson & Johnson
Acutely decompensated congestive heart failure; Cardiomyopathies; Cardiovascular Diseases; Coronary Disease; Diabetes Mellitus; Dyspnea; Heart Failure; Heart Failure, Systolic; Hyperemia; Hyperinsulinism; Hypertension; Myocardial Ischemia; Obesity; Renal Insufficiency; Sleep Disorders, Circadian Rhythm
Details
BaloncibartREGN-7544; REGN7544Phase 2 ClinicalRegeneron Pharmaceuticals Inc
Hypotension; Postural Orthostatic Tachycardia Syndrome
Details
XXB-750XXB-750Phase 2 ClinicalNovartis Pharma Ag
Heart Failure; Heart Failure, Systolic; Hypertension
Details
GNPPhase 2 ClinicalGuangzhou Leien Kangya Biomedical Technology Co Ltd
Acutely decompensated congestive heart failure; Heart Failure
Details
REGN-5381REGN-5381Phase 2 ClinicalRegeneron Pharmaceuticals Inc
Heart Failure; Hypertension
Details

Marketed Drug Information

English NameResearch CodeHighest Development StageCompanyFirst Brand NameFirst Approved CountryFirst IndicationFirst Approved CompanyFirst Approved DateIndicationClinical Trial
Recombinant human brain natriuretic peptide (Tibet Rhodiola)ApprovedTibet Rhodiola Pharmaceutical Holding Company新活素Mainland ChinaHeart FailureChengdu Rhodiola Bio-Pharmaceutical Co Ltd2005-04-11
Acutely decompensated congestive heart failure; Heart Failure
Details
Sodium NitroprussideSNPApprovedF. Hoffmann-La Roche LtdNipride, Nitriate, NitropressMainland ChinaHeart Failure; HypertensionChina Resources Double-Crane Pharmaceutical Co Ltd1974-05-10
Healthy Aging; Heart Failure; Hypertension; Hypotension; Myocardial Infarction; Pulmonary Edema; Schizophrenia
Details
Recombinant human brain natriuretic peptide (Suzhou Landing Bioteh)ApprovedSuzhou RxD Biopharmaceutical Co LtdMainland ChinaHeart FailureSuzhou RxD Biopharmaceutical Co Ltd2025-04-30
Heart Failure
Details
CarperitideSUN-Y4936r; alpha-hANP; ANF (99-126); SUN-4936r; ANP (99-126); CDD (99-126); SUN-4936; SUN-4936hApprovedDaiichi Sankyo Co LtdHANPJapanHeart FailureDaiichi Sankyo Co Ltd1995-01-20
Cardiomyopathies; Heart Failure; Respiratory Distress Syndrome, Adult
Details
Customer Reviews